nahso4-sio2: an efficient reusable green catalyst for selective c-3 propargylation of indoles with tertiary propargylic alcohols

نویسندگان

mukut gohani

johannes h. van tonder

barend c.b. benzuidenhoudt

چکیده

although several methods for the preparation of 4o propargyl indole derivatives have been published, this synthetic transformation is complicated by the tendency of 3o propargyl alcohols to form allenium intermediates in acidic media.  it is therefore a challenge to find an efficient method for the c-3 propargylation of indoles with 3° propargylic alcohols.  in this paper we wish to report on the successful application of silica gel impregnated with nahso4 as catalyst for the preparation of 4o propargyl indole derivatives.

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NaHSO4-SiO2: An Efficient Reusable Green Catalyst for Selective C-3 Propargylation of Indoles with Tertiary Propargylic Alcohols

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عنوان ژورنال:
iranian journal of chemistry and chemical engineering (ijcce)

ناشر: iranian institute of research and development in chemical industries (irdci)-acecr

ISSN 1021-9986

دوره 34

شماره 3 2015

میزبانی شده توسط پلتفرم ابری doprax.com

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